LEAD OPTIMIZATION
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GENEPEP offers its expertise in peptide chemistry for transforming your hits in lead compounds
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Through SAR studies, Genepep designs and synthesizes analogs of your molecule of interest for:
- Increasing stability, solubility, specificity and efficacy
- Reduce production cost
- Create new IP
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Structure-Activity studies
Identification of minimal active sequence, Ala scan, Gly-scan, D-scan, design of oriented libraries (analogs), incorporation of unnatural, exotic amino acid, peptide mimics, original cyclization …